Simon van der Plas

Publications by Year

Research Areas

Protein Kinase Regulation and GTPase Signaling, Synthesis and biological activity, Angiogenesis and VEGF in Cancer, Cancer, Hypoxia, and Metabolism, Immune cells in cancer

Most-Cited Works

• → Design, Synthesis, and Evaluation of Orally Active Benzimidazoles and Benzoxazoles as Vascular Endothelial Growth Factor-2 Receptor Tyrosine Kinase Inhibitors(2007)166 cited
• → The Role of the Acidity of N-Heteroaryl Sulfonamides as Inhibitors of Bcl-2 Family Protein–Protein Interactions(2013)73 cited
• → Allosteric Mutant IDH1 Inhibitors Reveal Mechanisms for IDH1 Mutant and Isoform Selectivity(2017)66 cited
• → Optimization of 3-Pyrimidin-4-yl-oxazolidin-2-ones as Allosteric and Mutant Specific Inhibitors of IDH1(2016)46 cited
• → Discovery of 2,4-bis-arylamino-1,3-pyrimidines as insulin-like growth factor-1 receptor (IGF-1R) inhibitors(2011)17 cited
• The role of the acidity of N-heteroaryl sulfonamides as inhibitors of Bcl-2 family protein-protein interactions(2013)