Karen Bresciano
Arqule (United States)(US)
Publications by Year
Research Areas
Computational Drug Discovery Methods, Pharmacogenetics and Drug Metabolism, PI3K/AKT/mTOR signaling in cancer, Protein Structure and Dynamics, Protein Kinase Regulation and GTPase Signaling
Most-Cited Works
- → Discovery and Optimization of a Series of 3-(3-Phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amines: Orally Bioavailable, Selective, and Potent ATP-Independent Akt Inhibitors(2012)99 cited
- → Characterization of a Phospholipase C β2-Binding Site Near the Amino-terminal Coiled-coil of G Protein βγ Subunits(2001)18 cited
- → Abstract 3231: In vitro cross species metabolism of a novel RAF kinase inhibitor phosphate prodrug, ARQ 736(2011)
- → Abstract C84: Nonclinical metabolism, disposition, pharmacokinetics, and in vitro drug-drug interaction assessment of ARQ 087, a pan-FGFR inhibitor.(2013)
- → Abstract 5783: In vitro ADME properties of ARQ 621: A specific Eg5 inhibitor(2010)
- → Abstract C83: Nonclinical in vitro ADME, disposition, and pharmacokinetic assessment of ARQ 092, a selective AKT inhibitor.(2013)