George Topalov
Publications by Year
Research Areas
Photoreceptor and optogenetics research, Enzyme function and inhibition, bioluminescence and chemiluminescence research, Synthesis and biological activity, Melanoma and MAPK Pathways
Most-Cited Works
- → Combinatorial computational method gives new picomolar ligands for a known enzyme(2002)78 cited
- → Potent and selective pyrazole-based inhibitors of B-Raf kinase(2008)65 cited
- → Non-oxime pyrazole based inhibitors of B-Raf kinase(2010)45 cited
- → Chlorophyll Catabolism Leading to the Skeleton of Dinoflagellate and Krill Luciferins: Hypothesis and Model Studies(2001)37 cited
- → Discovery of a Novel Class of Imidazo[1,2-a]Pyridines with Potent PDGFR Activity and Oral Bioavailability(2013)28 cited
- → Covalently cross-linked Watson–Crick base pair models. Part 2(2000)16 cited
- ARRY-334543, A potent, orally active small molecule inhibitor of EGFR and ErbB-2(2005)
- → Abstract 551: A potent and selective cFMS inhibitor regulates the tumor macrophage microenvironment leading to tumor growth inhibition(2011)1 cited
- → 303 Small molecule stabilizers of CFTR NBD1 can increase the protein half- life of the apical glycoform of F508del-CFTR to that of wild-type CFTR(2025)