Eric Boursier
Publications by Year
Research Areas
Protein Degradation and Inhibitors, RNA and protein synthesis mechanisms, Multiple Myeloma Research and Treatments, Chemical Synthesis and Analysis, Click Chemistry and Applications
Most-Cited Works
- → The bisindolylmaleimide GF 109203X is a potent and selective inhibitor of protein kinase C(1991)2,481 cited
- → Discovery and Characterization of Small Molecule Inhibitors of the BET Family Bromodomains(2011)334 cited
- → The Discovery of I-BET726 (GSK1324726A), a Potent Tetrahydroquinoline ApoA1 Up-Regulator and Selective BET Bromodomain Inhibitor(2014)187 cited
- → From ApoA1 upregulation to BET family bromodomain inhibition: Discovery of I-BET151(2012)118 cited
- → Discovery, SAR, and X-ray Binding Mode Study of BCATm Inhibitors from a Novel DNA-Encoded Library(2015)83 cited
- → Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors(2016)44 cited
- → The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits(2015)42 cited
- → Discovery of Pyridones As Oral AMPK Direct Activators(2013)14 cited
- → Abstract 782: Development of a high throughput in vitro screening platform to identify novel inducers of immunological cell death(2018)