Éric Malenfant
Boehringer Ingelheim (Canada)(CA)
Publications by Year
Research Areas
HIV Research and Treatment, HIV/AIDS drug development and treatment, Asymmetric Synthesis and Catalysis, Organoselenium and organotellurium chemistry, Axial and Atropisomeric Chirality Synthesis
Most-Cited Works
- → Discovery of BI 224436, a Noncatalytic Site Integrase Inhibitor (NCINI) of HIV-1(2014)176 cited
- → Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly(2010)104 cited
- → Asymmetric Ring Closure Reactions Mediated by a Chiral C2 Symmetrical Organoselenium Reagent(1995)91 cited
- → Peptidomimetic Inhibitors of the Human Cytomegalovirus Protease(1997)85 cited
- → Inhibition of Human Cytomegalovirus Protease by Monocyclic β-Lactam Derivatives: Kinetic Characterization Using a Fluorescent Probe(1999)74 cited
- → 2,6-Bis[(2S)-tetrahydrofuran-2-yl]phenyl diselenide: An effective reagent for asymmetric electrophilic addition reactions to olefins(1997)61 cited
- → Inhibition of human cytomegalovirus protease No with monocyclic β-lactams(1998)61 cited
- → Asymmetric arene-alkene cyclizations mediated by a chiral organoselenium reagent(1998)54 cited
- → Thiotetrazole alkynylacetanilides as potent and bioavailable non-nucleoside inhibitors of the HIV-1 wild type and K103N/Y181C double mutant reverse transcriptases(2007)53 cited
- → Novel Inhibitor Binding Site Discovery on HIV-1 Capsid N-Terminal Domain by NMR and X-ray Crystallography(2013)49 cited