Jason P. Burke
Publications by Year
Research Areas
Biochemical and Molecular Research, Cancer, Hypoxia, and Metabolism, Amino Acid Enzymes and Metabolism, Lung Cancer Treatments and Mutations, Protein Tyrosine Phosphatases
Most-Cited Works
- → Discovery of Small Molecules that Bind to K‐Ras and Inhibit Sos‐Mediated Activation(2012)495 cited
- → Discovery of Potent Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors Using Fragment-Based Methods and Structure-Based Design(2012)303 cited
- → Allosteric SHP2 Inhibitor, IACS-13909, Overcomes EGFR-Dependent and EGFR-Independent Resistance Mechanisms toward Osimertinib(2020)102 cited
- → Discovery of Tricyclic Indoles That Potently Inhibit Mcl-1 Using Fragment-Based Methods and Structure-Based Design(2015)95 cited
- → Discovery of IPN60090, a Clinical Stage Selective Glutaminase-1 (GLS-1) Inhibitor with Excellent Pharmacokinetic and Physicochemical Properties(2020)89 cited
- → Synthesis and Application of Chiral Cyclopropane-Based Ligands in Palladium-Catalyzed Allylic Alkylation(2004)80 cited
- → Branched polyesters: Preparative strategies and applications(2016)58 cited
- → Novel 2,3,4,5-tetrahydro-benzo[d]azepine derivatives of 2,4-diaminopyrimidine, selective and orally bioavailable ALK inhibitors with antitumor efficacy in ALCL mouse models(2010)34 cited
- → The Effect of Branching (Star Architecture) on Poly(d,l-lactide) (PDLLA) Degradation and Drug Delivery(2016)34 cited