M. Viļums
Leiden University(NL)Centre for Human Drug Research(NL)
Publications by Year
Research Areas
Synthesis and Characterization of Heterocyclic Compounds, Synthesis and biological activity, Chemokine receptors and signaling, Synthesis of heterocyclic compounds, Monoclonal and Polyclonal Antibodies Research
Most-Cited Works
- → Structure–Kinetic Relationships—An Overlooked Parameter in Hit-to-Lead Optimization: A Case of Cyclopentylamines as Chemokine Receptor 2 Antagonists(2013)61 cited
- → Discovery and Mapping of an Intracellular Antagonist Binding Site at the Chemokine Receptor CCR2(2014)54 cited
- → Indanes—Properties, Preparation, and Presence in Ligands for G Protein Coupled Receptors(2015)46 cited
- → When structure–affinity relationships meet structure–kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists(2015)26 cited
- → Synthesis, Cardiovascular Activity, and Electrochemical Oxidation of Nitriles of 5-Ethoxycarbonyl-2-methylthio-1,4-dihydropyridine-3-carboxylic Acid(2004)25 cited
- → Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E‐4031 Analogues(2011)19 cited
- → Cover Picture: Understanding of Molecular Substructures that Contribute to hERG K+ Channel Blockade: Synthesis and Biological Evaluation of E‐4031 Analogues (ChemMedChem 1/2012)(2011)9 cited
- → Evaluation of (4‐Arylpiperidin‐1‐yl)cyclopentanecarboxamides As High‐Affinity and Long‐Residence‐Time Antagonists for the CCR2 Receptor(2015)8 cited
- → Design and synthesis of novel small molecule CCR2 antagonists: Evaluation of 4-aminopiperidine derivatives(2014)8 cited
- → Alternative Products In One-Pot Reaction Of Benzylidene- Malononitrile, Thiocarbamoylacetamide And Alkyl Halides(2009)5 cited