Jacob A. Kaizerman
Publications by Year
Research Areas
Antibiotic Resistance in Bacteria, Cancer therapeutics and mechanisms, Antimicrobial Resistance in Staphylococcus, Bacteriophages and microbial interactions, Hedgehog Signaling Pathway Studies
Most-Cited Works
- → Potent and Highly Selective Hypoxia-Activated Achiral Phosphoramidate Mustards as Anticancer Drugs(2008)237 cited
- → DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 1: Internal benzimidazole derivatives(2004)128 cited
- → Discovery of AMG 925, a FLT3 and CDK4 Dual Kinase Inhibitor with Preferential Affinity for the Activated State of FLT3(2014)70 cited
- → DNA Binding Ligands Targeting Drug-Resistant Bacteria: Structure, Activity, and Pharmacology(2003)68 cited
- → DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 2: C-terminal benzimidazoles and derivatives(2004)56 cited
- → DNA Binding Ligands with Excellent Antibiotic Potency Against Drug-Resistant Gram-Positive Bacteria(2002)36 cited
- → Addressing PXR liabilities of phthalazine-based hedgehog/smoothened antagonists using novel pyridopyridazines(2010)32 cited
- → An Efficient and Scalable One-Pot Double Michael Addition-Dieckmann Condensation for the Synthesis of 4,4-Disubstituted Cyclohexane β-Keto Esters(2007)27 cited
- → DNA Binding Ligands with Improved in Vitro and in Vivo Potency against Drug-Resistant Staphylococcus aureus(2004)25 cited
- → Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors(2009)22 cited