Yann Dudit
GlaxoSmithKline (France)(FR)
Publications by Year
Research Areas
Protein Degradation and Inhibitors, Multiple Myeloma Research and Treatments, HIV Research and Treatment, Advanced biosensing and bioanalysis techniques, Diabetes Treatment and Management
Most-Cited Works
- → From ApoA1 upregulation to BET family bromodomain inhibition: Discovery of I-BET151(2012)118 cited
- → Naphthyridines as Novel BET Family Bromodomain Inhibitors(2013)34 cited
- → Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)(2016)20 cited
- → Discovery of Pyridones As Oral AMPK Direct Activators(2013)14 cited
- → The first bromodomain of human BRD4 in complex with 3,5 dimethylisoxaxole ligand(2013)