Jinshan M. Chen
Publications by Year
Research Areas
Ubiquitin and proteasome pathways, Click Chemistry and Applications, Synthesis and Catalytic Reactions, Protein Degradation and Inhibitors, Antibiotic Resistance in Bacteria
Most-Cited Works
- → Chemical and Computational Methods for the Characterization of Covalent Reactive Groups for the Prospective Design of Irreversible Inhibitors(2014)322 cited
- → Intrinsic reactivity profile of electrophilic moieties to guide covalent drug design: N-α-acetyl-l-lysine as an amine nucleophile(2016)63 cited
- → Binding site elucidation and structure guided design of macrocyclic IL-17A antagonists(2016)60 cited
- → Regulated induced proximity targeting chimeras—RIPTACs—A heterobifunctional small molecule strategy for cancer selective therapies(2024)55 cited
- → Heterocyclic methylsulfone hydroxamic acid LpxC inhibitors as Gram-negative antibacterial agents(2012)37 cited
- → Regulated Induced Proximity Targeting Chimeras (RIPTACs): a Novel Heterobifunctional Small Molecule Therapeutic Strategy for Killing Cancer Cells Selectively(2023)33 cited
- → Discovery and synthesis of novel 4-aminopyrrolopyrimidine Tie-2 kinase inhibitors for the treatment of solid tumors(2013)12 cited