J. Lépagnol
Université Libre de Bruxelles(BE)University of Liège(BE)AVL (France)(FR)Servier (France)(FR)
Publications by Year
Research Areas
Neuroscience and Neuropharmacology Research, Ion channel regulation and function, Nicotinic Acetylcholine Receptors Study, Phenothiazines and Benzothiazines Synthesis and Activities, Memory and Neural Mechanisms
Most-Cited Works
- → New Prolyl Endopeptidase Inhibitors: In Vitro and in Vivo Activities of Azabicyclo[2.2.2]octane, Azabicyclo[2.2.1]heptane, and Perhydroindole Derivatives(1996)90 cited
- → Structure−Activity Relationships in a Series of 2(1H)-Quinolones Bearing Different Acidic Function in the 3-Position: 6,7-Dichloro-2(1H)-oxoquinoline-3-phosphonic Acid, a New Potent and Selective AMPA/Kainate Antagonist with Neuroprotective Properties(1996)77 cited
- → 4H-1,2,4-Pyridothiadiazine 1,1-Dioxides and 2,3-Dihydro-4H-1,2,4-pyridothiadiazine 1,1-Dioxides Chemically Related to Diazoxide and Cyclothiazide as Powerful Positive Allosteric Modulators of (R/S)-2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors: Design, Synthesis, Pharmacology, and Structure−Activity Relationships(1998)60 cited
- → A new rapid method for phospholipid separation by high-performance liquid chromatography with light-scattering detection(1989)53 cited
- → Competitive inhibition by NBQX of kainate/AMPA receptor currents and excitatory synaptic potentials: importance of 6-nitro substitution(1992)51 cited