Rita Scarpelli
Italian Institute of Technology(IT)
Publications by Year
Research Areas
Cannabis and Cannabinoid Research, Histone Deacetylase Inhibitors Research, Synthetic Organic Chemistry Methods, Protein Degradation and Inhibitors, Peptidase Inhibition and Analysis
Most-Cited Works
- → Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection(2008)627 cited
- → Discovery of 2-{4-[(3S)-Piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): A Novel Oral Poly(ADP-ribose)polymerase (PARP) Inhibitor Efficacious in BRCA-1 and -2 Mutant Tumors(2009)308 cited
- → Structural and Functional Analysis of the Human HDAC4 Catalytic Domain Reveals a Regulatory Structural Zinc-binding Domain(2008)303 cited
- → Chemical synthesis and biological properties of pyridine epothilones(2000)144 cited
- → Multitarget Drug Discovery for Alzheimer's Disease: Triazinones as BACE‐1 and GSK‐3β Inhibitors(2014)122 cited
- → Dual inhibition of REV-ERBβ and autophagy as a novel pharmacological approach to induce cytotoxicity in cancer cells(2014)113 cited
- → Peripheral FAAH inhibition causes profound antinociception and protects against indomethacin-induced gastric lesions(2012)95 cited
- → Identification and Characterization of Carprofen as a Multitarget Fatty Acid Amide Hydrolase/Cyclooxygenase Inhibitor(2012)81 cited
- → Dihydroxypyrimidine-4-carboxamides as Novel Potent and Selective HIV Integrase Inhibitors(2007)76 cited
- → Discovery and Synthesis of HIV Integrase Inhibitors: Development of Potent and Orally Bioavailable N-Methyl Pyrimidones(2007)67 cited