Paul A. Stupple
Monash University(AU)
Publications by Year
Research Areas
Cyclopropane Reaction Mechanisms, Protein Degradation and Inhibitors, HIV/AIDS drug development and treatment, Synthesis and Catalytic Reactions, Cancer-related gene regulation
Most-Cited Works
- → Catalytic enantioselective rearrangements and cycloadditions involving ylides from diazo compounds(2001)334 cited
- → Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels(2013)241 cited
- → Subtype-Selective Small Molecule Inhibitors Reveal a Fundamental Role for Nav1.7 in Nociceptor Electrogenesis, Axonal Conduction and Presynaptic Release(2016)188 cited
- → HBO1 is required for the maintenance of leukaemia stem cells(2019)172 cited
- → Organocatalytic Asymmetric Total Synthesis of (R)-Rolipram and Formal Synthesis of (3S,4R)-Paroxetine(2008)147 cited
- → Regulation of PRMT5–MDM4 axis is critical in the response to CDK4/6 inhibitors in melanoma(2019)117 cited
- → Pyrazole NNRTIs 4: Selection of UK-453,061 (lersivirine) as a Development Candidate(2009)100 cited
- → Development of Dirhodium(II)-Catalyzed Generation and Enantioselective 1,3-Dipolar Cycloaddition of Carbonyl Ylides(2001)100 cited
- → Catalytic Enantioselective Tandem Carbonyl Ylide Formation-Cycloaddition(1997)94 cited
- → Discovery of Clinical Candidate 4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of NaV1.7(2017)83 cited