Linning Yu
Publications by Year
Research Areas
Estrogen and related hormone effects, Bioactive Compounds and Antitumor Agents, Pharmacogenetics and Drug Metabolism, Drug Transport and Resistance Mechanisms, Inflammatory mediators and NSAID effects
Most-Cited Works
- → Breast Cancer Resistance Protein (Bcrp/abcg2) Is a Major Determinant of Sulfasalazine Absorption and Elimination in the Mouse(2006)159 cited
- → Nuclear Magnetic Resonance Spectroscopy as a Quantitative Tool To Determine the Concentrations of Biologically Produced Metabolites: Implications in Metabolites in Safety Testing(2008)113 cited
- → Obtaining Exposures of Metabolites in Preclinical Species through Plasma Pooling and Quantitative NMR: Addressing Metabolites in Safety Testing (MIST) Guidance without Using Radiolabeled Compounds and Chemically Synthesized Metabolite Standards(2008)98 cited
- → Oxidation of Raloxifene to Quinoids: Potential Toxic Pathways via a Diquinone Methide and o-Quinones(2004)80 cited
- → Identification of Novel Electrophilic Metabolites of Piper methysticum Forst. (Kava)(2003)65 cited
- → Characterization of HKI-272 Covalent Binding to Human Serum Albumin(2010)60 cited
- → A Rational Chemical Intervention Strategy To Circumvent Bioactivation Liabilities Associated with a Nonpeptidyl Thrombopoietin Receptor Agonist Containing a 2-Amino-4-arylthiazole Motif(2007)51 cited
- → Synthesis and Reactivity of Potential Toxic Metabolites of Tamoxifen Analogues: Droloxifene and Toremifene o-Quinones(2001)35 cited
- → Bioactivation of Lamotrigine in Vivo in Rat and in Vitro in Human Liver Microsomes, Hepatocytes, and Epidermal Keratinocytes: Characterization of Thioether Conjugates by Liquid Chromatography/Mass Spectrometry and High Field Nuclear Magnetic Resonance Spectroscopy(2009)31 cited
- → Quinoids Formed from Estrogens and Antiestrogens(2004)29 cited