Mickaël Maudet

Publications by Year

Research Areas

Synthetic Organic Chemistry Methods, Carbohydrate Chemistry and Synthesis, PI3K/AKT/mTOR signaling in cancer, Traditional and Medicinal Uses of Annonaceae, Estrogen and related hormone effects

Most-Cited Works

• → Discovery of (R)-8-(1-(3,5-Difluorophenylamino)ethyl)-N,N-dimethyl-2-morpholino-4-oxo-4H-chromene-6-carboxamide (AZD8186): A Potent and Selective Inhibitor of PI3Kβ and PI3Kδ for the Treatment of PTEN-Deficient Cancers(2014)86 cited
• → Investigation of (E)-3-[4-(2-Oxo-3-aryl-chromen-4-yl)oxyphenyl]acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators(2015)42 cited
• → Asymmetric synthesis of (S)-(−)-N-acetylcolchinol via Ullmann biaryl coupling(2007)42 cited
• → Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors(2012)41 cited
• → New hydroxylamines for the synthesis of hydroxamic acids(1998)33 cited
• → Lignans.19. Total synthesis of (−)-O-dimethylsugiresinol, involving asymmetric [4+2] heterocycloaddition of a styrene with a benzylidenepyruvic ester of an α-O-silyl derivative of (D)-erythronolactone(1997)25 cited
• → High yield endoselective heterocycloadditions involving benzylidenepyruvic esters as the heterodiene and an alkoxystyrene as the dienophile(1994)23 cited
• → Strategic studies in the syntheses of novel 6,7-substituted quinolones and 7- or 6-substituted 1,6- and 1,7-naphthyridones(2008)22 cited
• → An efficient large-scale synthesis of alkyl 5-hydroxy-pyridin- and pyrimidin-2-yl acetate(2008)22 cited
• → Asymmetric endoselective [4+2] heterocycloadditions of styrene dienophiles with chiral benzylidenepyruvic esters. Total synthesis of (−)-O-dimethylsugiresinol(1997)21 cited