Rui‐Yang Yang
Arqule (United States)(US)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Asymmetric Synthesis and Catalysis, Synthesis and Catalytic Reactions, Fluorine in Organic Chemistry, Cancer therapeutics and mechanisms
Most-Cited Works
- → Discovery and Optimization of a Series of 3-(3-Phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amines: Orally Bioavailable, Selective, and Potent ATP-Independent Akt Inhibitors(2012)99 cited
- → Solution and solid phase synthesis of 5-alkoxyhydantoin libraries with a three-fold functional diversity(1996)86 cited
- → The asymmetric synthesis of allylglycine and other unnatural α-amino acids via zinc-mediated allylation of oximes in aqueous media(1996)81 cited
- → Synthetic methods for the preparation of ARQ 501 (β-Lapachone) human blood metabolites(2008)58 cited
- → A concise and efficient solid-phase synthesis of 2-amino-4(3H)-quinazolinones(2000)51 cited
- → Enantioselective allylation of α-ketoester oximes with an external chiral ligand: Asymmetric synthesis of allylglycines and allylalanine(1996)50 cited
- → Asymmetric synthesis of L-azetidine-2-carboxylic acid and 3-substituted congeners—conformationally constrained analogs of phenylalanine, naphthylalanine, and leucine(1999)42 cited
- → Zinc-Mediated Allylation of N-Protected α-Amino Aldehydes in Aqueous Solution. Stereoselective Synthesis of Phe-Phe Hydroxyethylene Dipeptide Isosteres(1997)36 cited
- → Zinc-Mediated Allylation of N-Protected α-Amino Aldehydes in Aqueous Solution. Stereoselective Synthesis of Anti- and Syn-β-Amino Alcohols with Functionalized Allyl Groups(1997)36 cited
- → Synthesis of cyclic iodonium ylides—3H-1λ3-benziodol-1-ylium ylides via transylidation of iodonium ylides to iodides(1992)32 cited