George M. Burslem
Kaiser Permanente(US)California University of Pennsylvania(US)Institute of Biophysics(BG)University of Pennsylvania(US)Epigenomics (Germany)(DE)
Publications by Year
Research Areas
Protein Degradation and Inhibitors, Ubiquitin and proteasome pathways, Peptidase Inhibition and Analysis, Click Chemistry and Applications, Chemical Synthesis and Analysis
Most-Cited Works
- → Proteolysis-Targeting Chimeras as Therapeutics and Tools for Biological Discovery(2020)974 cited
- → Lessons in PROTAC Design from Selective Degradation with a Promiscuous Warhead(2017)876 cited
- → The Advantages of Targeted Protein Degradation Over Inhibition: An RTK Case Study(2017)650 cited
- → Small-Molecule Modulation of Protein Homeostasis(2017)285 cited
- → Targeting BCR-ABL1 in Chronic Myeloid Leukemia by PROTAC-Mediated Targeted Protein Degradation(2019)217 cited
- → Enhancing Antiproliferative Activity and Selectivity of a FLT-3 Inhibitor by Proteolysis Targeting Chimera Conversion(2018)170 cited