Stefano Crosignani
Galderma (Switzerland)(CH)
Publications by Year
Research Areas
Tryptophan and brain disorders, Chemical Synthesis and Analysis, Adenosine and Purinergic Signaling, Chemical Synthesis and Reactions, Nanoplatforms for cancer theranostics
Most-Cited Works
- → Discovery of a Novel and Selective Indoleamine 2,3-Dioxygenase (IDO-1) Inhibitor 3-(5-Fluoro-1H-indol-3-yl)pyrrolidine-2,5-dione (EOS200271/PF-06840003) and Its Characterization as a Potential Clinical Candidate(2017)135 cited
- → Discovery of a New Class of Potent, Selective, and Orally Bioavailable CRTH2 (DP2) Receptor Antagonists for the Treatment of Allergic Inflammatory Diseases(2008)103 cited
- → Characterization of the Selective Indoleamine 2,3-Dioxygenase-1 (IDO1) Catalytic Inhibitor EOS200271/PF-06840003 Supports IDO1 as a Critical Resistance Mechanism to PD-(L)1 Blockade Therapy(2018)83 cited
- → Inhibition of Tryptophan-Dioxygenase Activity Increases the Antitumor Efficacy of Immune Checkpoint Inhibitors(2019)68 cited
- → Optimization of the Central Core of Indolinone–Acetic Acid-Based CRTH2 (DP2) Receptor Antagonists(2011)64 cited
- → Polymer-Supported Mukaiyama Reagent: A Useful Coupling Reagent for the Synthesis of Esters and Amides(2004)62 cited
- → Chiral amplification in Diels-Alder and 1,3-dipolar cycloadditions catalyzed by bis(oxazoline)-Zn(II)-based chiral complexes(1999)60 cited
- → Novel Application of α-Azido Aldehydes in Multicomponent Reactions: Synthesis of Triazolo-Fused Dihydrooxazinones via a Passerini Reaction–Dipolar Cycloaddition Strategy(2011)48 cited
- → 4-Naphthyl-substituted bis(oxazoline): A new, easily recoverable and efficient chiral ligand in asymmetric catalysis of the Diels-Alder reaction(1998)47 cited
- → Polymer-Supported O-Alkylisoureas: Useful Reagents for the O-Alkylation of Carboxylic Acids(2004)37 cited