Paul S. Humphries
California Department of Public Health(US)
Publications by Year
Research Areas
Peroxisome Proliferator-Activated Receptors, Chemical synthesis and alkaloids, Asymmetric Synthesis and Catalysis, Metabolism, Diabetes, and Cancer, Adipose Tissue and Metabolism
Most-Cited Works
- → Carbazole-containing sulfonamides and sulfamides: Discovery of cryptochrome modulators as antidiabetic agents(2015)74 cited
- → Carbazole-containing amides and ureas: Discovery of cryptochrome modulators as antihyperglycemic agents(2017)51 cited
- → Synthesis and SAR of 1,2,3,4-tetrahydroisoquinolin-1-ones as novel G-protein-coupled receptor 40 (GPR40) antagonists(2009)51 cited
- → Structure-based design of novel human Pin1 inhibitors (III): Optimizing affinity beyond the phosphate recognition pocket(2014)49 cited
- → Microwave-assisted synthesis utilizing supported reagents: a rapid and versatile synthesis of 1,5-diarylpyrazoles(2006)47 cited
- → The discovery of novel calcium sensing receptor negative allosteric modulators(2009)41 cited
- → A Formal Asymmetric Synthesis of (+)-Anatoxin-a Using an Enantioselective Deprotonation Strategy on an Eight-Membered Ring(1999)39 cited
- → Synthesis and SAR of 4-substituted-2-aminopyrimidines as novel c-Jun N-terminal kinase (JNK) inhibitors(2009)26 cited
- → Pyrimidone-based series of glucokinase activators with alternative donor–acceptor motif(2013)22 cited
- → Enantioselective deprotonation of 4-tert-butylcyclohexanone by conformationally constrained chiral lithium amide bases(1999)21 cited