Christopher Housseman
Publications by Year
Research Areas
Computational Drug Discovery Methods, Asymmetric Synthesis and Catalysis, Chemical Synthesis and Analysis, Cancer Mechanisms and Therapy, Multicomponent Synthesis of Heterocycles
Most-Cited Works
- → The Enantioselective Morita–Baylis–Hillman Reaction and Its Aza Counterpart(2007)480 cited
- → Discovery of 2-[[2-Ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2- a ]pyridin-3-yl]methylamino]-4-(4-fluorophenyl)thiazole-5-carbonitrile (GLPG1690), a First-in-Class Autotaxin Inhibitor Undergoing Clinical Evaluation for the Treatment of Idiopathic Pulmonary Fibrosis(2017)137 cited
- → Enantioselektive Morita‐Baylis‐Hillman‐Reaktionen und ihre Aza‐Varianten(2007)98 cited
- → Discovery, Structure–Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors(2017)60 cited
- → Identification of a 4-(Hydroxymethyl)diarylhydantoin as a Selective Androgen Receptor Modulator(2012)51 cited
- → Mono Alkylation of α-Isocyano Acetamide to its Higher Homologues(2006)9 cited
- → Synthesis of α-Isocyano-α-alkyl(aryl)acetamides and their Use in the Multicomponent Synthesis of 5-Aminooxazole, Pyrrolo[3,4-b]pyridin-5-one and 4,5,6,7-Tetrahydrofuro[2,3-c]pyridine(2004)7 cited
- → Synthesis of α‐Isocyano‐α‐alkyl(aryl)acetamides and Their Use in the Multicomponent Synthesis of 5‐Aminooxazole, Pyrrolo[3,4‐b]pyridin‐5‐one and 4,5,6,7‐Tetrahydrofuro[2,3‐c]pyridine.(2005)6 cited
- → Monoalkylation of α‐Isocyano Acetamide to Its Higher Homologues.(2006)2 cited
- → Abstract 4191: Combining artificial intelligence and human expertise in pursuit of novel PolQ inhibitors(2025)1 cited