Andrew B. Hague
Infinity Pharmaceuticals (United States)(US)
Publications by Year
Research Areas
Organic and Inorganic Chemical Reactions, Asymmetric Synthesis and Catalysis, Fluorine in Organic Chemistry, Marine Sponges and Natural Products, Advanced Synthetic Organic Chemistry
Most-Cited Works
- → Discovery of a Potent, Orally Active 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor for Clinical Study: Identification of (S)-2-((1S,2S,4R)-Bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one (AMG 221)(2010)80 cited
- → A One-Pot Tandem Pictet-Spengler-Diels-Alder Synthesis of Apoyohimbines from 3-Carbomethoxy-2-(formylmethyl)-3-sulfolene(1997)21 cited
- → Development of a Multi Kilogram-Scale, Tandem Cyclopropanation Ring-Expansion Reaction en Route to Hedgehog Antagonist IPI-926(2016)9 cited
- → (4-Piperidinylphenyl)aminoethyl amides as a novel class of non-covalent cathepsin K inhibitors(2003)8 cited
- → The Geometry of Dienes from 2,3-Substituted-3-Sulfolenes and the Stereoselectivity of their Intramolecular Diels-Alder Cyclisations(1997)6 cited
- → Interesting stereoselectivity of intramolecular Diels-Alder reactions leading to 5-carbomethoxy yohimbine systems(1999)4 cited
- → Chapter 6 Preparation of substituted 3-sulfolenes and their use as precursors for diels-alder dienes(1998)4 cited
- → A Practical Large-Scale Synthesis of 3-Carbomethoxy-3-sulfolene(2000)3 cited
- → ChemInform Abstract: Preparation of Substituted 3‐Sulfolenes and Their Use as Precursors for Diels—Alder Dienes(1998)
- → ChemInform Abstract: A Practical Large‐Scale Synthesis of 3‐Carbomethoxy‐3‐sulfolene.(2000)