Thomas E. Barta
Johannes Kepler University of Linz(AT)
Publications by Year
Research Areas
Peptidase Inhibition and Analysis, Lipid Membrane Structure and Behavior, Protease and Inhibitor Mechanisms, Heat shock proteins research, Computational Drug Discovery Methods
Most-Cited Works
- → Discovery of Novel 2-Aminobenzamide Inhibitors of Heat Shock Protein 90 as Potent, Selective and Orally Active Antitumor Agents(2009)189 cited
- → Small molecule inhibitors of Hsp90 potently affect inflammatory disease pathways and exhibit activity in models of rheumatoid arthritis(2008)134 cited
- → Orally Active MMP-1 Sparing α-Tetrahydropyranyl and α-Piperidinyl Sulfone Matrix Metalloproteinase (MMP) Inhibitors with Efficacy in Cancer, Arthritis, and Cardiovascular Disease(2010)97 cited
- → Discovery of benzamide tetrahydro-4H-carbazol-4-ones as novel small molecule inhibitors of Hsp90(2008)89 cited
- → Application of Chemoproteomics to Drug Discovery: Identification of a Clinical Candidate Targeting Hsp90(2010)87 cited
- → Stereocontrol in the intramolecular Diels-Alder reaction. 7. Use of the trimethylsilyl group as a removable stereocontrol element to provide greatly enhanced levels of diastereoselection(1985)77 cited
- → Synthesis and Structure−Activity Relationships of β- and α-Piperidine Sulfone Hydroxamic Acid Matrix Metalloproteinase Inhibitors with Oral Antitumor Efficacy(2005)64 cited
- → Antiinflammatory 4,5-diarylimidazoles as selective cyclooxygenase inhibitors(1998)60 cited
- → Fluorescence Linked Enzyme Chemoproteomic Strategy for Discovery of a Potent and Selective DAPK1 and ZIPK Inhibitor(2013)49 cited
- → Quantification of Water Flux in Vesicular Systems(2018)44 cited