K. Jeff Thrasher
Eli Lilly (United States)(US)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Synthesis and Reactions of Organic Compounds, Estrogen and related hormone effects, Synthesis and Catalytic Reactions, Quinazolinone synthesis and applications
Most-Cited Works
- → Discovery and Synthesis of [6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]- 2-(4-hydroxyphenyl)]benzo[b]thiophene: A Novel, Highly Potent, Selective Estrogen Receptor Modulator(1997)176 cited
- → Quinazolinone cholecystokinin-B receptor ligands(1991)63 cited
- → Dibasic Benzo[b]thiophene Derivatives as a Novel Class of Active Site-Directed Thrombin Inhibitors. 1. Determination of the Serine Protease Selectivity, Structure−Activity Relationships, and Binding Orientation(1997)54 cited
- → Phenothiazines as lipid peroxidation inhibitors and cytoprotective agents(1992)45 cited
- → Discovery of N-(6-Fluoro-1-oxo-1,2-dihydroisoquinolin-7-yl)-5-[(3R)-3-hydroxypyrrolidin-1-yl]thiophene-2-sulfonamide (LSN 3213128), a Potent and Selective Nonclassical Antifolate Aminoimidazole-4-carboxamide Ribonucleotide Formyltransferase (AICARFT) Inhibitor Effective at Tumor Suppression in a Cancer Xenograft Model(2017)33 cited
- → Structural Evolution and Pharmacology of a Novel Series of Triacid Angiotensin II Receptor Antagonists(1994)24 cited
- → Characterization of a novel AICARFT inhibitor which potently elevates ZMP and has anti-tumor activity in murine models(2018)20 cited
- → Chiral recognition of the angiotensin II (AT1) receptor by a highly potent phenoxyproline octanoamide(1994)10 cited
- → Quinoline-substituted dihydroindoles as cysLT1 (LTD4 receptor) antagonists(1996)8 cited
- → Pyridine Metallations in the Synthesis of Triazole Based NK-1 Antagonists(2006)7 cited