Dalia R. Jakas
South College(US)GlaxoSmithKline (United States)(US)
Publications by Year
Research Areas
Cell Adhesion Molecules Research, Synthesis and biological activity, Cancer therapeutics and mechanisms, Synthesis and Reactions of Organic Compounds, Glycosylation and Glycoproteins Research
Most-Cited Works
- → Synthesis of water-soluble (aminoalkyl)camptothecin analogs: inhibition of topoisomerase I and antitumor activity(1991)516 cited
- → Modification of the hydroxylactone ring of camptothecin: inhibition of mammalian topoisomerase I and biological activity(1989)411 cited
- → Indole Naphthyridinones as Inhibitors of Bacterial Enoyl-ACP Reductases FabI and FabK(2003)161 cited
- → Defining and Combating the Mechanisms of Triclosan Resistance in Clinical Isolates ofStaphylococcus aureus(2002)96 cited
- → Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists(1996)72 cited
- → Conformational Preferences in a Benzodiazepine Series of Potent Nonpeptide Fibrinogen Receptor Antagonists(1999)53 cited
- → Semisynthetic cephalosporins. Synthesis and structure-activity relations of 7-mandelamido-3-cephem-4-carboxylic acids(1974)46 cited
- → Preclinical Pharmacokinetics and Interspecies Scaling of a Novel Vitronectin Receptor Antagonist(1999)39 cited
- → Orally bioavailable nonpeptide vitronectin receptor antagonists with efficacy in an osteoporosis model(1999)35 cited
- → Orally active 7-phenylglycyl cephalosporins. Structure-activity studies related to cefatrizine (SK&F 60771).(1976)33 cited