Vinayak Hosagrahara
Publications by Year
Research Areas
Peroxisome Proliferator-Activated Receptors, Tuberculosis Research and Epidemiology, Pharmacogenetics and Drug Metabolism, Drug Transport and Resistance Mechanisms, Cancer therapeutics and mechanisms
Most-Cited Works
- → Raising HDL cholesterol without inducing hepatic steatosis and hypertriglyceridemia by a selective LXR modulator(2004)186 cited
- → Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo(2013)161 cited
- → Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis(2017)124 cited
- → Epoxide hydrolase — polymorphism and role in toxicology(2000)121 cited
- → 4-Aminoquinolone Piperidine Amides: Noncovalent Inhibitors of DprE1 with Long Residence Time and Potent Antimycobacterial Activity(2014)94 cited
- → Discovery of Pyrazolopyridones as a Novel Class of Noncovalent DprE1 Inhibitor with Potent Anti-Mycobacterial Activity(2014)93 cited
- → Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate(2015)73 cited
- → Reactivity of mefenamic acid 1-o-acyl glucuronide with proteins in vitro and ex vivo.(1996)65 cited
- → Identification of Orally Available Naphthyridine Protein Kinase D Inhibitors(2010)53 cited
- → Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279(2023)51 cited