David E. Coppa
Novartis (United States)(US)
Publications by Year
Research Areas
Protease and Inhibitor Mechanisms, Peptidase Inhibition and Analysis, Oral microbiology and periodontitis research, Inflammatory mediators and NSAID effects, Monoclonal and Polyclonal Antibodies Research
Most-Cited Works
- → Identification of Dipeptidyl Nitriles as Potent and Selective Inhibitors of Cathepsin B through Structure-Based Drug Design(2001)136 cited
- → N-Arylaminonitriles as bioavailable peptidomimetic inhibitors of cathepsin B(2003)28 cited
- → Carboxy-Substituted Cinnamides: A Novel Series of Potent, Orally Active LTB4 Receptor Antagonists(1998)20 cited
- → Cathepsin B complexed with dipeptidyl nitrile inhibitor(2001)