Kshitij Thakkar
La Roche College(US)
Publications by Year
Research Areas
Cancer Treatment and Pharmacology, Oxidative Organic Chemistry Reactions, Traditional and Medicinal Uses of Annonaceae, Synthesis of Organic Compounds, Asymmetric Synthesis and Catalysis
Most-Cited Works
- → Discovery of 2-[3,5-Dichloro-4-(5-isopropyl-6-oxo-1,6-dihydropyridazin-3-yloxy)phenyl]-3,5-dioxo-2,3,4,5-tetrahydro[1,2,4]triazine-6-carbonitrile (MGL-3196), a Highly Selective Thyroid Hormone Receptor β Agonist in Clinical Trials for the Treatment of Dyslipidemia(2014)208 cited
- → Synthesis and protein-tyrosine kinase inhibitory activity of polyhydroxylated stilbene analogs of piceatannol(1993)145 cited
- → A Novel Oxidative Cyclization of 2'-Hydroxychalcones to 4,5-Dialkoxyaurones by Thallium(III) Nitrate(1995)74 cited
- → Preparation and Diastereoselective Birch Reduction−Alkylation of Chiral 3,4-Dihydro-1(2H)-isoquinolinones. Enantiospecific Syntheses and Opioid Receptor Affinities of Several Hydro-2,3- dimethyl-1H-7,12a-methanobenzo[6,7]cycloocta[1,2-c]pyridine-9-ols(1998)30 cited
- → A novel oxidative cyclization of 2′-hydroxychalcones to 4-methoxyaurones by thallium (III) nitrate(1994)29 cited
- → 7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: Novel and highly selective protein tyrosine phosphatase 1B inhibitors(2012)22 cited
- → Discovery of a Highly Potent, Orally Active Mitosis/Angiogenesis Inhibitor R1530 for the Treatment of Solid Tumors(2013)22 cited
- → Novel Fragmentation Reaction of 2-Alkyl- and 2,4-Dialkyl-3-iodo-1-oxocyclohexan-2,4-carbolactones(2004)21 cited
- → Asymmetric synthesis and fragmentation reactions of 2-alkyl- and 2, 4-dialkyl-3-iodo-1-oxocyclohexan-2, 4-carbolactones. Single enantiomer preparation of Δα, β-butenolides, 2-alkyl-4-hydroxy-2-cyclohexen-1-ones and butyrolactones(1998)17 cited
- → Pyrazolobenzodiazepines: Part I. Synthesis and SAR of a potent class of kinase inhibitors(2010)14 cited