Leonard D. Rodman
United States Military Academy(US)
Publications by Year
Research Areas
HER2/EGFR in Cancer Research, Angiogenesis and VEGF in Cancer, Cancer Treatment and Pharmacology, Quinazolinone synthesis and applications, PI3K/AKT/mTOR signaling in cancer
Most-Cited Works
- → Potent N-(1,3-Thiazol-2-yl)pyridin-2-amine Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors with Excellent Pharmacokinetics and Low Affinity for the hERG Ion Channel(2004)60 cited
- → The discovery of N-(1,3-thiazol-2-yl)pyridin-2-amines as potent inhibitors of KDR kinase(2004)36 cited
- → Potent 2-[(pyrimidin-4-yl)amine}-1,3-thiazole-5-carbonitrile-based inhibitors of VEGFR-2 (KDR) kinase(2005)35 cited
- → 2,4-Disubstituted pyrimidines: A novel class of KDR kinase inhibitors(2003)28 cited
- → 2,4‐Disubstituted Pyrimidines: A Novel Class of KDR Kinase Inhibitors.(2003)1 cited
- Development of 3-methylpyridin-2-yl-aminothiazole inhibitors of the VEGF receptor(2003)