Melissa S. Egbertson
Egis (France)(FR)
Publications by Year
Research Areas
Platelet Disorders and Treatments, HIV/AIDS drug development and treatment, Biochemical and Molecular Research, HIV Research and Treatment, Antiplatelet Therapy and Cardiovascular Diseases
Most-Cited Works
- → Diketo acid inhibitor mechanism and HIV-1 integrase: Implications for metal binding in the active site of phosphotransferase enzymes(2002)395 cited
- → A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase(2004)332 cited
- → HIV-1 integrase inhibitors that compete with the target DNA substrate define a unique strand transfer conformation for integrase(2000)317 cited
- → Non-peptide fibrinogen receptor antagonists. 1. Discovery and design of exosite inhibitors(1992)295 cited
- → Design and Synthesis of 8-Hydroxy-[1,6]Naphthyridines as Novel Inhibitors of HIV-1 Integrase in Vitro and in Infected Cells(2003)268 cited
- → 4-Aryl-2,4-dioxobutanoic Acid Inhibitors of HIV-1 Integrase and Viral Replication in Cells(2000)187 cited
- → Non-Peptide Fibrinogen Receptor Antagonists. 2. Optimization of a Tyrosine Template as a Mimic for Arg-Gly-Asp(1994)178 cited
- → Maximizing Diversity from a Kinase Screen: Identification of Novel and Selective pan-Trk Inhibitors for Chronic Pain(2014)60 cited
- → The characterization of intermediates in the mitomycin activation cascade: a practical synthesis of an aziridinomitosene(1986)55 cited
- → Non-Peptide GPIIb/IIIa Inhibitors. 20. Centrally Constrained Thienothiophene α-Sulfonamides Are Potent, Long Acting in Vivo Inhibitors of Platelet Aggregation(1999)50 cited