Bheemarao G. Ugarkar
AstraZeneca (India)(IN)
Publications by Year
Research Areas
Biochemical and Molecular Research, Adenosine and Purinergic Signaling, HIV/AIDS drug development and treatment, Quinazolinone synthesis and applications, Phenothiazines and Benzothiazines Synthesis and Activities
Most-Cited Works
- → Design, Synthesis, and Characterization of a Series of Cytochrome P4503A-Activated Prodrugs (HepDirect Prodrugs) Useful for Targeting Phosph(on)ate-Based Drugs to the Liver§(2004)157 cited
- → Adenosine Kinase Inhibitors. 1. Synthesis, Enzyme Inhibition, and Antiseizure Activity of 5-Iodotubercidin Analogues(2000)111 cited
- → Adenosine Kinase Inhibitors as a Novel Approach to Anticonvulsant Therapy(1999)99 cited
- → Quinolinyl Pyrimidines: Potent Inhibitors of NDH-2 as a Novel Class of Anti-TB Agents(2012)93 cited
- → Pradefovir: A Prodrug That Targets Adefovir to the Liver for the Treatment of Hepatitis B(2008)73 cited
- → Discovery of benzothiazoles as antimycobacterial agents: Synthesis, structure–activity relationships and binding studies with Mycobacterium tuberculosis decaprenylphosphoryl-β-d-ribose 2′-oxidase(2015)58 cited
- → Adenosine Kinase Inhibitors. 6. Synthesis, Water Solubility, and Antinociceptive Activity of 5-Phenyl-7-(5-deoxy-β-d-ribofuranosyl)pyrrolo[2,3-d]pyrimidines Substituted at C4 with Glycinamides and Related Compounds(2005)58 cited
- → Adenosine Kinase Inhibitors. 2. Synthesis, Enzyme Inhibition, and Antiseizure Activity of Diaryltubercidin Analogues(2000)53 cited
- → Structure Guided Lead Generation for M. tuberculosis Thymidylate Kinase (Mtb TMK): Discovery of 3-Cyanopyridone and 1,6-Naphthyridin-2-one as Potent Inhibitors(2014)44 cited
- → Synthesis and Characterization of a Novel Liver-Targeted Prodrug of Cytosine-1-β-d-arabinofuranoside Monophosphate for the Treatment of Hepatocellular Carcinoma(2006)44 cited