Thea Mulder‐Krieger
Leiden University(NL)Centre for Human Drug Research(NL)
Publications by Year
Research Areas
Adenosine and Purinergic Signaling, Receptor Mechanisms and Signaling, Pharmacological Receptor Mechanisms and Effects, Synthesis and Biological Evaluation, Neuropeptides and Animal Physiology
Most-Cited Works
- → Functional efficacy of adenosine A2Areceptor agonists is positively correlated to their receptor residence time(2012)185 cited
- → New, Non-Adenosine, High-Potency Agonists for the Human Adenosine A2B Receptor with an Improved Selectivity Profile Compared to the Reference Agonist N-Ethylcarboxamidoadenosine(2004)150 cited
- → Predicting Binding Affinities for GPCR Ligands Using Free-Energy Perturbation(2016)145 cited
- → 2-Amino-6-furan-2-yl-4-substituted Nicotinonitriles as A2A Adenosine Receptor Antagonists(2008)144 cited
- → A Series of Ligands Displaying a Remarkable Agonistic−Antagonistic Profile at the Adenosine A1 Receptor(2004)114 cited
- → 2,4,6-Trisubstituted Pyrimidines as a New Class of Selective Adenosine A1 Receptor Antagonists(2004)94 cited
- → Dual-Point Competition Association Assay: A Fast and High-Throughput Kinetic Screening Method for Assessing Ligand-Receptor Binding Kinetics(2012)65 cited
- → A Series of 2,4-Disubstituted Quinolines as a New Class of Allosteric Enhancers of the Adenosine A3Receptor(2009)63 cited
- → Identifying Novel Adenosine Receptor Ligands by Simultaneous Proteochemometric Modeling of Rat and Human Bioactivity Data(2012)53 cited
- → The endocannabinoid 2-arachidonylglycerol is a negative allosteric modulator of the human A3 adenosine receptor(2009)50 cited