Ronald J. Mattson
Bristol-Myers Squibb (United States)(US)
Publications by Year
Research Areas
Neurotransmitter Receptor Influence on Behavior, Synthesis and Biological Evaluation, Stress Responses and Cortisol, Receptor Mechanisms and Signaling, Asymmetric Synthesis and Catalysis
Most-Cited Works
- → An improved method for reductive alkylation of amines using titanium(IV) isopropoxide and sodium cyanoborohydride(1990)185 cited
- → Enantioselective Synthesis of a Highly Potent Selective Serotonin Reuptake Inhibitor. An Application of Imidazolidinone Catalysis to the Alkylation of Indoles with an α,β-Disubstituted α,β-Unsaturated Aldehyde(2005)123 cited
- → A Strategy to Minimize Reactive Metabolite Formation: Discovery of (S)-4-(1-Cyclopropyl-2-methoxyethyl)-6-[6-(difluoromethoxy)-2,5-dimethylpyridin-3-ylamino]-5-oxo-4,5-dihydropyrazine-2-carbonitrile as a Potent, Orally Bioavailable Corticotropin-Releasing Factor-1 Receptor Antagonist(2009)54 cited
- → [3H]5-carboxamidotryptamine labels multiple high affinity 5-HT1D-like sites in guinea pig brain(1991)46 cited
- → Conformationally restricted homotryptamines 3. Indole tetrahydropyridines and cyclohexenylamines as selective serotonin reuptake inhibitors(2007)40 cited
- → Ortho-directed lithiation in .pi.-deficient diazinyl heterocycles(1990)40 cited
- → In Vitro Intrinsic Clearance-Based Optimization ofN3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists(2009)38 cited
- → Aminotriazine 5-HT7 antagonists(2004)36 cited
- → Catalytic Asymmetric Diazoacetate Cyclopropanation of 1-Tosyl-3-vinylindoles. A Route to Conformationally Restricted Homotryptamines(2005)36 cited
- → Conformationally Restricted Homotryptamines. 2. Indole Cyclopropylmethylamines as Selective Serotonin Reuptake Inhibitors(2005)33 cited