Ronald Wolin
Janssen (United States)(US)
Publications by Year
Research Areas
Protein Kinase Regulation and GTPase Signaling, Chemical Synthesis and Analysis, Mast cells and histamine, Oxidative Organic Chemistry Reactions, Asymmetric Synthesis and Catalysis
Most-Cited Works
- → Novel pyrazole derivatives as potent inhibitors of type II topoisomerases. Part 1: Synthesis and preliminary SAR analysis(2007)99 cited
- → (+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]- pyridin-11(R)-yl)-1-piperidinyl]-2-oxo-ethyl]-1-piperidinecarboxamide (SCH-66336): A Very Potent Farnesyl Protein Transferase Inhibitor as a Novel Antitumor Agent(1998)97 cited
- → Electroreductive cyclization. Ketones and aldehydes tethered to .alpha.,.beta.-unsaturated esters (nitriles). Fundamental investigations(1988)67 cited
- → New Sequential Carbon-Carbon Bond Forming Reactions. A Samarium(II) Iodide Mediated Vinylogous Barbier Reaction Followed by an Aldol Reaction(1991)63 cited
- → Synthesis and evaluation of pyrazolo[3,4-b]quinoline ribofuranosides and their derivatives as inhibitors of oncogenic Ras(1996)57 cited
- → Electroreductive cyclization reactions. Stereoselection, creation of quaternary centers in bicyclic frameworks, and a formal total synthesis of quadrone.(1990)56 cited
- → Discovery and SAR of 6-Alkyl-2,4-diaminopyrimidines as Histamine H4 Receptor Antagonists(2014)37 cited
- → Pyrrolidino-tetrahydroisoquinolines as potent dual H3 antagonist and serotonin transporter inhibitors(2007)31 cited
- → Triaryl bis-sulfones as cannabinoid-2 receptor ligands: SAR studies(2005)28 cited
- → A novel B-RAF inhibitor blocks interleukin-8 (IL-8) synthesis in human melanoma xenografts, revealing IL-8 as a potential pharmacodynamic biomarker(2008)27 cited