Donald F. Worth
Publications by Year
Research Areas
Synthesis and Characterization of Heterocyclic Compounds, Synthesis and biological activity, Synthesis and Biological Evaluation, Chemical Reaction Mechanisms, Synthesis of heterocyclic compounds
Most-Cited Works
- → 1-Substituted 7-[3-[(ethylamino)methyl]-1-pyrrolidinyl]-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids. New quantitative structure activity relationships at N1 for the quinolone antibacterials(1988)96 cited
- → Laboratory Studies on 4,6-Diamino-1-(p-Chlorophenyl)-1,2-Dihydro-2,2-Dimethyl-s-Triazine Pamoate (CI-501) as a Repository Antimalarial Drug(1963)61 cited
- → Synthesis of xanthines as adenosine antagonists, a practical quantitative structure-activity relationship application(1985)60 cited
- → Antimalarial drugs. 60. Synthesis, antimalarial activity, and quantitative structure-activity relationships of tebuquine and a series of related 5-[(7-chloro-4-quinolinyl)amino]-3-[(alkylamino)methyl][1,1'-biphenyl]-2-ols and N.omega.-oxides(1986)52 cited
- → Synthesis and structure-activity relationships of pyrazolo[4,3-d]pyrimidin-7-ones as adenosine receptor antagonists(1987)49 cited
- → 1,4‐Cyeloaddition reactions. IV. preparation of Cyclopenta[g]furo[3,2‐c]quinolines, Cyclopenta‐ [f]furo[3,2‐c]quinolines, Benzo[H]furo[3,2‐c]quinolines, and Furo‐ [3,2‐c]indeno[1,7‐gh] quinolines from 2,3‐Dihydro‐5‐methylfuran and schiff bases(1970)35 cited
- → Repository drugs. IV. 4',4'''-Sulfonylbisacetanilide (acedapsone, DADDS) and related sulfanilylanilides with prolonged antimalarial and antileprotic action(1969)34 cited
- → Antimalarial drugs. 25. Folate antagonists. 3. 2,4-Diamino-6-(heterocyclic)quinazolines, a novel class of antimetabolites with potent antimalarial and antibacterial activity(1972)32 cited
- → Basically substituted ellipticine analogs as potential antitumor agents(1986)29 cited
- → Antimalarial drugs. 39. Folate antagonists. 13. 2,4-Diamino-6-[(.alpha.,.alpha.,.alpha.-trifluoro-m-tolyl)thio]quinazoline and related 2,4-diamino-6-[(phenyl- and naphthyl)thio]quinazolines, a unique class of antimetabolites with extraordinary antimalarial and antibacterial effects(1978)28 cited