Michael S. Hadley
Icahn School of Medicine at Mount Sinai(US)
Publications by Year
Research Areas
Receptor Mechanisms and Signaling, Asymmetric Synthesis and Catalysis, Synthesis of heterocyclic compounds, Synthesis and Biological Evaluation, Phenothiazines and Benzothiazines Synthesis and Activities
Most-Cited Works
- → Pharmacological Actions of a Novel, High-Affinity, and Selective Human Dopamine D3 Receptor Antagonist, SB-277011-A(2000)288 cited
- → Comparison of azabicyclic esters and oxadiazoles as ligands for the muscarinic receptor(1991)204 cited
- → 1,3-Biarylureas as selective non-peptide antagonists of the orexin-1 receptor(2001)165 cited
- → Design and Synthesis of trans-N-[4-[2-(6-Cyano-1,2,3,4-tetrahydroisoquinolin-2- yl)ethyl]cyclohexyl]-4-quinolinecarboxamide (SB-277011): A Potent and Selective Dopamine D3 Receptor Antagonist with High Oral Bioavailability and CNS Penetration in the Rat(2000)129 cited
- → Design and Synthesis oftrans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1H-3-benzazepine (SB-414796): A Potent and Selective Dopamine D3Receptor Antagonist(2003)72 cited
- → Synthesis and antihypertensive activity of 3-[(substituted-carbonyl)amino]-2H-1-benzopyrans