Fuk‐Wah Sum
Publications by Year
Research Areas
NF-κB Signaling Pathways, Peptidase Inhibition and Analysis, Pancreatic and Hepatic Oncology Research, Receptor Mechanisms and Signaling, Pharmacological Effects and Assays
Most-Cited Works
- → 5-Fluoro-2-methyl-N-[4-(5H-pyrrolo[2,1-c]- [1,4]benzodiazepin-10(11H)-ylcarbonyl)-3- chlorophenyl]benzamide (VPA-985): An Orally Active Arginine Vasopressin Antagonist with Selectivity for V2Receptors(1998)148 cited
- → Stereoselective synthesis of β-substituted α,β-unsaturated esters by dialkylcuprate coupling to the enol phosphate of β-keto esters(1979)105 cited
- → Indole Cytosolic Phospholipase A2α Inhibitors: Discovery and in Vitro and in Vivo Characterization of 4-{3-[5-Chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic Acid, Efipladib(2008)88 cited
- → Inhibition of Cytosolic Phospholipase A2α: Hit to Lead Optimization(2005)76 cited
- → Novel (4-Piperidin-1-yl)-phenyl Sulfonamides as Potent and Selective Human β3 Agonists(2001)45 cited
- → 2,4-thiazolidinediones as potent and selective human β3 agonists(2001)43 cited
- → Structure–activity study of novel tricyclic benzazepine arginine vasopressin antagonists(2003)41 cited
- → Structure-Activity Relationship of 6-Methylidene Penems Bearing 6,5 Bicyclic Heterocycles as Broad-Spectrum β-Lactamase Inhibitors: Evidence for 1,4-Thiazepine Intermediates with C7 R Stereochemistry by Computational Methods(2006)40 cited
- → Cyclic amine sulfonamides as linkers in the design and synthesis of novel human β3 adrenergic receptor agonists(2003)22 cited
- → (4-Piperidin-1-yl)phenyl Amides: Potent and Selective Human β3 Agonists(2001)22 cited