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2(S)-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine (1): A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor Antagonist

Journal of Medicinal Chemistry1996Vol. 39(9), pp. 1760–1762

Citations Over TimeTop 16% of 1996 papers

Jeffrey J. Hale, Sander G. Mills, Malcolm MacCoss, Shrenik K. Shah, Hongbo Qi, David J. Mathre, Margaret A. Cascieri, Sharon Sadowski, Catherine D. Strader, D. Euan MacIntyre, Joseph M. Metzger

Abstract

ADVERTISEMENT RETURN TO ISSUEPREVLetterNEXT2(S)-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3(S)-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine (1): A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor AntagonistJeffrey J. Hale, Sander G. Mills, Malcolm MacCoss, Shrenik K. Shah, Hongbo Qi, David J. Mathre, Margaret A. Cascieri, Sharon Sadowski, Catherine D. Strader, D. Euan MacIntyre, and Joseph M. MetzgerView Author Information Merck Research Laboratories, Rahway, New Jersey 07065Cite this: J. Med. Chem. 1996, 39, 9, 1760–1762Publication Date (Web):April 26, 1996Publication History Received1 September 1995Published online26 April 1996Published inissue 1 January 1996https://pubs.acs.org/doi/10.1021/jm950654whttps://doi.org/10.1021/jm950654wrapid-communicationACS PublicationsCopyright © 1996 American Chemical SocietyRequest reuse permissionsArticle Views1229Altmetric-Citations63LEARN ABOUT THESE METRICSArticle Views are the COUNTER-compliant sum of full text article downloads since November 2008 (both PDF and HTML) across all institutions and individuals. These metrics are regularly updated to reflect usage leading up to the last few days.Citations are the number of other articles citing this article, calculated by Crossref and updated daily. Find more information about Crossref citation counts.The Altmetric Attention Score is a quantitative measure of the attention that a research article has received online. Clicking on the donut icon will load a page at altmetric.com with additional details about the score and the social media presence for the given article. Find more information on the Altmetric Attention Score and how the score is calculated. Share Add toView InAdd Full Text with ReferenceAdd Description ExportRISCitationCitation and abstractCitation and referencesMore Options Share onFacebookTwitterWechatLinked InRedditEmail Other access optionsGet e-AlertscloseSupporting Info (1)»Supporting Information Supporting Information SUBJECTS:Antagonists,Calcium,Molecular structure,Piperidines,Receptors Get e-Alerts

Citations Over TimeTop 16% of 1996 papers

Abstract

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