N→S Acyl-Transfer-Mediated Synthesis of Peptide Thioesters Using Anilide Derivatives
Organic Letters2009Vol. 11(4), pp. 823–826
Citations Over TimeTop 10% of 2009 papers
Abstract
N-->S acyl-transfer-mediated synthesis of peptide thioesters utilizing an N-aminoacyl-N-sulfanylethylaminobenzoic acid derivative has been examined. The developed synthetic methodology for peptide thioesters is compatible with Fmoc solid-phase peptide synthesis (SPPS).
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