Optimization of triazole-based TGR5 agonists towards orally available agents
MedChemComm2012Vol. 4(1), pp. 205–210
Citations Over TimeTop 17% of 2012 papers
Kentaro Futatsugi, Kevin B. Bahnck, Martin Brenner, Joanne Buxton, Janice E. Chin, Steven B. Coffey, Jeffrey S. Dubins, Declan Flynn, Denise Gautreau, Angel Guzmán-Pérez, John R. Hadcock, David Hepworth, Michael Herr, Terri Hinchey, Ann M. Janssen, Sandra M. Jennings, Wenhua Jiao, Sophie Y. Lavergne, Bryan Li, Mei Li, Michael J. Munchhof, Suvi T. M. Orr, David W. Piotrowski, Nicole Roush, M. F. Sammons, Benjamin D. Stevens, Gregory Storer, Jian Wang, Joseph S. Warmus, Liuqing Wei, Angela Wolford
Abstract
With the challenge of striking the balance of TGR5 potency and clearance, the screening strategy as well as medicinal chemistry strategy are discussed in this article.
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