Benoı̂t Laleu
Medicines for Malaria Venture(CH)
Publications by Year
Research Areas
Malaria Research and Control, Computational Drug Discovery Methods, HIV/AIDS drug development and treatment, Crystallization and Solubility Studies, X-ray Diffraction in Crystallography
Most-Cited Works
- → Nicotinamide adenine dinucleotide phosphate oxidase in experimental liver fibrosis: GKT137831 as a novel potential therapeutic agent(2012)335 cited
- → First in Class, Potent, and Orally Bioavailable NADPH Oxidase Isoform 4 (Nox4) Inhibitors for the Treatment of Idiopathic Pulmonary Fibrosis(2010)234 cited
- → Exploiting the Divergent Reactivity of Aryl–Palladium Intermediates for the Rapid Assembly of Fluorene and Phenanthrene Derivatives(2009)174 cited
- → A Palladium-Catalyzed Alkylation/Direct Arylation Synthesis of Nitrogen-Containing Heterocycles(2008)99 cited
- → Resolution of [4]Heterohelicenium Dyes with Unprecedented Pummerer‐like Chemistry(2005)86 cited
- → Synthesis of Annulated 2H-Indazoles and 1,2,3- and 1,2,4-Triazoles via a One-Pot Palladium-Catalyzed Alkylation/Direct Arylation Reaction(2008)85 cited
- → Design, synthesis and biological activity of original pyrazolo-pyrido-diazepine, -pyrazine and -oxazine dione derivatives as novel dual Nox4/Nox1 inhibitors(2011)78 cited
- → Screening of the ‘Pathogen Box’ identifies an approved pesticide with major anthelmintic activity against the barber's pole worm(2016)75 cited
- → The Development Process for Discovery and Clinical Advancement of Modern Antimalarials(2019)73 cited
- → Screening of TB Actives for Activity against Nontuberculous Mycobacteria Delivers High Hit Rates(2017)71 cited