Andrew Ayscough
University of Cambridge(GB)
Publications by Year
Research Areas
Peptidase Inhibition and Analysis, Synthesis and Catalytic Reactions, Crystallization and Solubility Studies, X-ray Diffraction in Crystallography, Quinazolinone synthesis and applications
Most-Cited Works
- → CHR-2797: An Antiproliferative Aminopeptidase Inhibitor that Leads to Amino Acid Deprivation in Human Leukemic Cells(2008)117 cited
- → Assessing molecular scaffolds for CNS drug discovery(2017)56 cited
- → Structure–activity relationships of the peptide deformylase inhibitor BB-3497: modification of the methylene spacer and the P1′ side chain(2003)33 cited
- → 1,2,4-Triazolo-[1,5-a]pyridine HIF Prolylhydroxylase Domain-1 (PHD-1) Inhibitors With a Novel Monodentate Binding Interaction(2017)33 cited
- → Peptide Deformylase Inhibitors, Potential for a New Class of Broad Spectrum Antibacterials(2002)27 cited
- → Structure–activity relationships of the peptide deformylase inhibitor BB-3497: modification of the P2′ and P3′ side chains(2003)27 cited
- → Synthesis of a simplified analogue of eleutherobin via a Claisen rearrangement and ring closing metathesis strategy(2005)20 cited
- → Diastereoselective aziridination of alkenes using 3-acetoxyamino-2-(1-hydroxyalkyl)quinazolin-4(3H )-ones in the presence of titanium(IV) tert-butoxide(1998)18 cited
- → Conformational diastereoisomers of PPh3 coordinated to stereogenic metal centres as molecular optical switches(2001)16 cited
- → Reagent- and chelation-controlled diastereoselective aziridination of electron-rich alkenes by 3-acetoxyamino-2-(1-hydroxy-2,2-dimethylprop-1-yl)-quinazolin-4(3H)-one(1996)15 cited