Amrita Bobok
Gedeon Richter (Hungary)(HU)
Publications by Year
Research Areas
Pharmacological Receptor Mechanisms and Effects, Neuroscience and Neuropharmacology Research, Receptor Mechanisms and Signaling, Neurotransmitter Receptor Influence on Behavior, Nicotinic Acetylcholine Receptors Study
Most-Cited Works
- → Neuronal Dopamine D3 Receptors: Translational Implications for Preclinical Research and CNS Disorders(2021)67 cited
- → Poster #16 CARIPRAZINE, A D3/D2 DOPAMINE RECEPTOR PARTIAL AGONIST ANTIPSYCHOTIC, DISPLAYS GREATER D3 RECEPTOR OCCUPANCY IN VIVO COMPARED WITH OTHER ANTIPSYCHOTICS(2012)30 cited
- → In vitro and in vivo comparison of [3H](+)‐PHNO and [3H]raclopride binding to rat striatum and lobes 9 and 10 of the cerebellum: A method to distinguish dopamine D3from D2receptor sites: A method to distinguish dopamine D3from D2receptor sites(2010)29 cited
- → Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications(2017)29 cited
- → 4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate(2016)21 cited
- → Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists(2010)21 cited
- → Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs(2010)20 cited
- → Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization(2015)15 cited
- → Cell-based and virtual fragment screening for adrenergic α2C receptor agonists(2015)11 cited
- → Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization(2014)11 cited