Taegyo Lee
Pfizer (United States)(US)
Publications by Year
Research Areas
Catalytic C–H Functionalization Methods, Asymmetric Hydrogenation and Catalysis, Cyclopropane Reaction Mechanisms, Computational Drug Discovery Methods, Catalytic Cross-Coupling Reactions
Most-Cited Works
- → Rhodium-Catalyzed Enantioselective Silylation of Arene C–H Bonds: Desymmetrization of Diarylmethanols(2015)125 cited
- → Rhodium‐Catalyzed Enantioselective Silylation of Cyclopropyl C−H Bonds(2016)119 cited
- → Iridium-Catalyzed, β-Selective C(sp3)–H Silylation of Aliphatic Amines To Form Silapyrrolidines and 1,2-Amino Alcohols(2018)92 cited
- → Highly Modular Synthesis of 1,2-Diketones via Multicomponent Coupling Reactions of Isocyanides as CO Equivalents(2019)46 cited
- → Mechanistic Studies on Rhodium-Catalyzed Enantioselective Silylation of Aryl C–H Bonds(2017)43 cited
- → Development of the Commercial Manufacturing Process for Nirmatrelvir in 17 Months(2023)37 cited
- → Synthesis of Nirmatrelvir: Development of a Scalable Cobalt-Catalyzed Cyclopropanation for Manufacture of the Bicyclic [3.1.0]Proline-Building Block(2023)19 cited
- → S N Ar Regioselectivity Predictions: Machine Learning Triggering DFT Reaction Modeling through Statistical Threshold(2023)15 cited
- → Synthesis of Nirmatrelvir: Design and Optimization of an Efficient Telescoped Amidation–Dehydration Sequence(2023)14 cited