Gareth W. Harbottle
Publications by Year
Research Areas
Prostate Cancer Treatment and Research, Asymmetric Synthesis and Catalysis, Cancer, Lipids, and Metabolism, Protein Degradation and Inhibitors, Chemical Synthesis and Analysis
Most-Cited Works
- → Targeting the p300/CBP Axis in Lethal Prostate Cancer(2021)271 cited
- → Cycloaddition of Chiral tert-Butanesulfinimines with Trimethylenemethane(2013)36 cited
- → Convergent Asymmetric Synthesis of Two Complex TRPV1 Antagonists(2011)27 cited
- → Characterisation of CCS1477: A novel small molecule inhibitor of p300/CBP for the treatment of castration resistant prostate cancer.(2017)24 cited
- → Structure–activity relationships of novel non-competitive mGluR1 antagonists: A potential treatment for chronic pain(2006)21 cited
- → In vitro and in vivo SAR of pyrido[3,4-d]pyramid-4-ylamine based mGluR1 antagonists(2009)17 cited
- → Selective fluorination of 1-hydroxyisoquinolines using Selectfluor™(2007)14 cited
- → Microwave-assisted synthesis of mGluR1 ligands: carbon, nitrogen and oxygen linked derivatives of pyrido[3,4-d]pyrimidin-4-ylamines(2007)12 cited
- → Two-directional synthesis and biological evaluation of alkaloid 5-epi-cis-275B′(2014)6 cited
- → Combining Two-Directional Synthesis and Tandem Reactions, Part 17: Expedient Formation of Functionalised Azabicycles(2012)2 cited