Attila Bielik
Gedeon Richter (Hungary)(HU)
Publications by Year
Research Areas
Neuroscience and Neuropharmacology Research, Chemical Synthesis and Analysis, Pharmacological Receptor Mechanisms and Effects, Quinazolinone synthesis and applications, Synthesis of heterocyclic compounds
Most-Cited Works
- → A High Throughput Luminescent Assay for Glycogen Synthase Kinase-3 β Inhibitors(2007)121 cited
- → Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists(2003)36 cited
- → Discovery and Preclinical Characterization of 3-((4-(4-Chlorophenyl)-7-fluoroquinoline-3-yl)sulfonyl)benzonitrile, a Novel Non-acetylenic Metabotropic Glutamate Receptor 5 (mGluR5) Negative Allosteric Modulator for Psychiatric Indications(2017)29 cited
- → Novel sulfonamides having dual dopamine D2 and D3 receptor affinity show in vivo antipsychotic efficacy with beneficial cognitive and EPS profile(2007)21 cited
- → Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists(2010)21 cited
- → Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs(2010)20 cited
- → Novel solid-phase synthesis of 2,6-disubstituted 4(3H)-quinazolinones for combinatorial library generation(2002)19 cited
- → Solid-phase synthesis of 6-hydroxy-2,4-diaminoquinazolines(2005)14 cited
- → Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu 5 ) receptor negative allosteric modulators(2017)9 cited
- → Scheduling a Flexible, Open-Architecture Robotic Workstation under LabWindows(2005)8 cited