Elena Casale
Institut National de Recherche pour l'Agriculture, l'Alimentation et l'Environnement(FR)Toxalim Research Centre in Food Toxicology(FR)
Publications by Year
Research Areas
Heat shock proteins research, Computational Drug Discovery Methods, Quinazolinone synthesis and applications, Synthesis and biological activity, Chronic Myeloid Leukemia Treatments
Most-Cited Works
- → The target landscape of clinical kinase drugs(2017)850 cited
- → Through the “Gatekeeper Door”: Exploiting the Active Kinase Conformation(2009)502 cited
- → Covalent and allosteric inhibitors of the ATPase VCP/p97 induce cancer cell death(2013)381 cited
- → 3-Aminopyrazole Inhibitors of CDK2/Cyclin A as Antitumor Agents. 1. Lead Finding(2004)159 cited
- → Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy(2015)141 cited
- → Crystal Structure of the T315I Abl Mutant in Complex with the Aurora Kinases Inhibitor PHA-739358(2007)132 cited