Randall J. Gallaschun
Publications by Year
Research Areas
Synthesis and pharmacology of benzodiazepine derivatives, Stress Responses and Cortisol, Hormonal Regulation and Hypertension, Computational Drug Discovery Methods, Synthesis and biological activity
Most-Cited Works
- → Inhibition of the oncogene product p185erbB-2 in vitro and in vivo by geldanamycin and dihydrogeldanamycin derivatives(1995)199 cited
- → erbB-2 oncogene inhibition by geldanamycin derivatives: synthesis, mechanism of action, and structure-activity relationships(1995)138 cited
- → Treatment with HC-070, a potent inhibitor of TRPC4 and TRPC5, leads to anxiolytic and antidepressant effects in mice(2018)136 cited
- → Synthesis and Oral Efficacy of a 4-(Butylethylamino)pyrrolo[2,3-d]pyrimidine: A Centrally Active Corticotropin-Releasing Factor1 Receptor Antagonist(1997)113 cited
- → 2-Aryloxy-4-alkylaminopyridines: Discovery of Novel Corticotropin-Releasing Factor 1 Antagonists(2008)69 cited
- → Synthesis and SAR of 2-Aryloxy-4-alkoxy-pyridines as Potent Orally Active Corticotropin-Releasing Factor 1 Receptor Antagonists(2008)48 cited
- → Discovery and Characterization of a Novel Dihydroisoxazole Class of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) Receptor Potentiators(2013)22 cited
- → Quantitative structure-activity relationships of antitumor guanidinothiazolecarboxamides with survival enhancement for therapy in the 3LL Lewis lung carcinoma model(1991)12 cited
- → Synthesis of 1,2-dihydro-1-oxo-3H-3-benzazepine and 3-acyl derivatives(1989)11 cited
- → Synthesis of novel 1,3‐oxazino[6,5‐b]indole‐2,4‐(3H,9H)‐dione and 2H‐1,3,5‐oxadiazino[3,2‐a]indole‐2,4‐(3H)‐dione from oxindoles(1992)10 cited