Steve Keeling
Publications by Year
Research Areas
Cyclization and Aryne Chemistry, Chemical Synthesis and Analysis, Asymmetric Synthesis and Catalysis, Synthesis and Biological Evaluation, Synthetic Organic Chemistry Methods
Most-Cited Works
- → New Synthesis of 1-Substituted-1H-indazoles via 1,3-Dipolar Cycloaddition of in situ Generated Nitrile Imines and Benzyne(2010)153 cited
- → An improved synthesis of 1,2-benzisoxazoles: TBAF mediated 1,3-dipolar cycloaddition of nitrile oxides and benzyne(2010)59 cited
- → Addressing species specific metabolism and solubility issues in a quinoline series of oral PDE4 inhibitors(2009)35 cited
- → An efficient entry to 1,2-benzisoxazoles via 1,3-dipolar cycloaddition of in situ generated nitrile oxides and benzyne(2010)34 cited
- → Pyrrolidinones derived from (S )-pyroglutamic acid. Part 1. Conformationally constrained glutamate(2000)31 cited
- → Pyrrolidinones derived from (S )-pyroglutamic acid. Part 2. Conformationally constrained kainoid analogues(2000)29 cited
- → Optimization of Orally Bioavailable PI3Kδ Inhibitors and Identification of Vps34 as a Key Selectivity Target(2019)18 cited
- → Functionalised pyrrolidinones by conjugate addition of stabilised enolates and Reformatsky reagents(1996)17 cited
- → Direct versatile route to conformationally constrained glutamate analogues(1998)14 cited
- → Discovery of a potent series of non-steroidal non α-trifluoromethyl carbinol glucocorticoid receptor agonists with reduced lipophilicity(2011)8 cited