Simon Surprenant
Aegera Therapeutics (Canada)(CA)
Publications by Year
Research Areas
Chemical Synthesis and Analysis, Synthetic Organic Chemistry Methods, Asymmetric Synthesis and Catalysis, Click Chemistry and Applications, Chemical Synthesis and Reactions
Most-Cited Works
- → Systematic Study of the Synthesis of Macrocyclic Dipeptide β-Turn Mimics Possessing 8-, 9-, and 10- Membered Rings by Ring-Closing Metathesis(2005)85 cited
- → Efficient Synthesis of Substituted Vinyl Ethers Using the Julia Olefination(2003)56 cited
- → From Macrocycle Dipeptide Lactams To Azabicyclo[X.Y.0]alkanone Amino Acids: A Transannular Cyclization Route for Peptide Mimic Synthesis(2006)36 cited
- → Inhibition of HIV-1 capsid assembly: Optimization of the antiviral potency by site selective modifications at N1, C2 and C16 of a 5-(5-furan-2-yl-pyrazol-1-yl)-1H-benzimidazole scaffold(2012)35 cited
- → Efficient Nucleophilic Aromatic Substitution between Aryl Nitrofluorides and Alkynes(2007)30 cited
- → Aligning Potency and Pharmacokinetic Properties for Pyridine-Based NCINIs(2016)23 cited
- → 9-(4-Bromophenyl)-9-fluorenyl as a Safety-Catch Nitrogen Protecting Group(2005)9 cited
- → Systematic Study of the Synthesis of Macrocyclic Dipeptide β-Turn Mimics Possessing 8-, 9-, and 10-Membered Rings by Ring-Closing Metathesis.(2005)9 cited
- → Discovery of RP-1664: A First-in-Class Orally Bioavailable, Selective PLK4 Inhibitor(2025)8 cited
- → The Discovery of RP-2119: A Potent, Selective, and Orally Bioavailable Polθ ATPase Inhibitor(2025)7 cited